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Front MatterAbstract - Hi-Res PDF (727 KB) - PDF w/links (728 KB)
Chapter 1. Screening of Endogenous Ligands for Orphan GPCRsTetsuya Ohtaki, Masahiko Fujino, Shuji Hinuma, Masaaki MoriAbstract - Hi-Res PDF (2638 KB) - PDF w/links (1784 KB)
Chapter 2. Screening of Ligands for Human GPCRs by the Use of Receptor-G alpha Fusion ProteinsHinako SugaAbstract - Hi-Res PDF (867 KB) - PDF w/links (886 KB)
Chapter 3. Screening and Identification of Ghrelin, an Endogenous Ligand for GHS-RKenji Kangawa, Masayasu KojimaAbstract - Hi-Res PDF (715 KB) - PDF w/links (735 KB)
Chapter 4. Ligand Screening of Olfactory ReceptorsTakao Nakagawa, Kazushige Touhara, Sayako Katada, Yuki OkaAbstract - Hi-Res PDF (1487 KB) - PDF w/links (1519 KB)
Chapter 5. Generation and Phenotypical Analysis of Muscarinic Acetylcholine Receptor Knockout MiceChuxia Deng, Sung-Jun Han, Jongrye Jeon, Cuiling Li, Dinesh Gautam, Jürgen WessAbstract - Hi-Res PDF (883 KB) - PDF w/links (749 KB)
Chapter 6. Systematic Mutagenesis of M1 Muscarinic Acetylcholine ReceptorsEdward C. HulmeAbstract - Hi-Res PDF (2020 KB) - PDF w/links (1193 KB)
Chapter 7. Analysis of the Regulation of Muscarinic Acetylcholine ReceptorsChris J. van KoppenAbstract - Hi-Res PDF (579 KB) - PDF w/links (584 KB)
Chapter 8. Single-Molecule Analysis of Chemotactic Signaling Mediated by cAMP Receptor on Living CellsYukihiro Miyanaga, Toshio Yanagida, Masahiro UedaAbstract - Hi-Res PDF (1966 KB) - PDF w/links (930 KB)
Chapter 9. Oligomerization of G Protein-Coupled Purinergic ReceptorsHiroyasu Nakata, Kazuaki Yoshioka, Toshio KamiyaAbstract - Hi-Res PDF (1260 KB) - PDF w/links (918 KB)
Chapter 10. Methods and Results in X-Ray Crystallography of Bovine RhodopsinRumi Tsujimoto, Chihiro Funamoto, Tetsuji Okada, Miho MuraokaAbstract - Hi-Res PDF (1821 KB) - PDF w/links (847 KB)
Chapter 11. Determination of Steric Structure of Muscarinic Ligands Bound to Muscarinic Acetylcholine ReceptorsMasaji Ishiguro, Toshiyuki Hamada, Hiroshi Hirota, Hiroyasu FurukawaAbstract - Hi-Res PDF (1640 KB) - PDF w/links (869 KB)
Chapter 12. Modeling of G Protein-Coupled Receptors for Drug DesignMasaji IshiguroAbstract - Hi-Res PDF (2142 KB) - PDF w/links (978 KB)
Color InsertAbstract - Hi-Res PDF (2528 KB) - PDF w/links (546 KB)