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Front MatterAbstract - Hi-Res PDF (448 KB) - PDF w/links (449 KB)
Chapter 1. IntroductionAbstract - Hi-Res PDF (306 KB) - PDF w/links (307 KB)
Chapter 2. Biology of G Protein-Coupled ReceptorsAbstract - Hi-Res PDF (573 KB) - PDF w/links (585 KB)
Chapter 3. G Protein-Coupled Receptors as Targets for Drug DiscoveryTimothy A. EsbenshadeAbstract - Hi-Res PDF (1046 KB) - PDF w/links (1068 KB)
Chapter 4. G Protein-Coupled Receptors as Cardiovascular Drug TargetsAmir Snapir, Mika ScheininAbstract - Hi-Res PDF (918 KB) - PDF w/links (926 KB)
Chapter 5. G Protein-Coupled Receptors and CancerRemko A. Bakker, Martine J. SmitAbstract - Hi-Res PDF (985 KB) - PDF w/links (794 KB)
Chapter 6. G Protein-Coupled Receptors in Metabolic DiseaseRegina M. Reilly, Christine A. CollinsAbstract - Hi-Res PDF (546 KB) - PDF w/links (579 KB)
Chapter 7. G Protein-Coupled Receptors in CNS Drug DiscoveryRita Raddatz, Deborah S. HartmanAbstract - Hi-Res PDF (767 KB) - PDF w/links (796 KB)
Chapter 8. Recombinant G Protein-Coupled Receptors for Drug DiscoveryAbstract - Hi-Res PDF (528 KB) - PDF w/links (547 KB)
Chapter 9. High Throughput Screening Assays for G Protein-Coupled ReceptorsDavid Burns, Sujatha Gopalakrishnan, Jurgen Vanhauwe, Usha WarriorAbstract - Hi-Res PDF (668 KB) - PDF w/links (689 KB)
Chapter 10. Molecular Bioinformatics of Receptor Binding and ActivationHeike Obermann, Kevan P. Willey, James B. ProcterAbstract - Hi-Res PDF (3474 KB) - PDF w/links (2204 KB)
Chapter 11. Structures and Dynamics of G Protein-Coupled ReceptorsJudith Klein-Seetharaman, Michèle C. LoewenAbstract - Hi-Res PDF (1765 KB) - PDF w/links (1670 KB)
Chapter 12. Toward Crystallization of G Protein-Coupled ReceptorsMaria P. MacWilliamsAbstract - Hi-Res PDF (1807 KB) - PDF w/links (1611 KB)
Chapter 13. Novel Solid-State NMR Methods for Structural Studies on G Protein-Coupled ReceptorsAdam Lange, Marc BaldusAbstract - Hi-Res PDF (1980 KB) - PDF w/links (1090 KB)
Chapter 14. Structural Genomics InitiativesKenneth H LundstromAbstract - Hi-Res PDF (525 KB) - PDF w/links (533 KB)
Chapter 15. Molecular Basis of Dimerization of Family A G Protein-Coupled ReceptorsGraeme MilliganAbstract - Hi-Res PDF (412 KB) - PDF w/links (427 KB)
Chapter 16. Orphan ReceptorsOlivier Civelli, Yumiko Saito, Zhiwei WangAbstract - Hi-Res PDF (565 KB) - PDF w/links (586 KB)